(4R,6R)-tert-Butyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxan-4-acetat CAS NO.{{ 10}}

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(4R,6R)-tert-Butyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxan-4-acetat CAS NO.{{ 10}}
Detaljer
MF: C14H23NO4
MW: 269,34
Einecs:425-780-3
Produkt klassificering
Atorvastatin mellemprodukter
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(4R,6R)-tert-butyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxan-4-acetat Grundlæggende oplysninger

produktnavn (4R,6R)-tert-butyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxan-4-acetat
Synonymer ATS-8;(4R,6R)-T-BUTYL-6-CYANOMETHYL-2,2-DIMETHYL-1,3-DIOXAN{{10} }ACETATE;(4R,6R)-TERT-BUTYL-6-CYANOMETHYL-2,2-DIMETHYL-1,3-DIOXAN-4-ACETATE;( 4R,CIS)-1,1-DIMETHYLETHYL-6-CYANOMETHYL-2,2-DIMETHYL-1,3-DIOXAN{{29} }ACETATE;(4R,3R)-TERT-BUTYL-6-CYANOMETHYL-2,2-DIMETHYL-1,3-DIOXAN-4-ACETATE;( 4R-CIS)-1,1-DIMETHYLETHYL-6-CYANOMETHYL-2,2-DIMETHYL-1,3-DIOXAN{{49} }ACETAT (ATS-8);tert-Butyl (4R,3R)-6-cyanomethyl-2,2-dimethyl-1,3-dioxan{ {59}}acetat;TERT-BUTYL[(4R,6R)-6-CYANOMETHYL-2,2-DIMETHYL-1,3-DIOXAN-4- YL]ACETAT
CAS 125971-94-0
MF C14H23NO4
MW 269.34
Einecs-nummer 425-780-3

 

(4R,6R)-tert-butyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxan-4-acetat Kemiske egenskaber

Smeltepunkt 65-69 grad (belyst)
Kogepunkt 364,1±17.0 grader (forudsagt)
massefylde 1.016±0,06 g/cm3(forudsagt)
opbevarings temp. 2-8 grad
opløselighed opløseligt i chloroform
formular pulver til krystal
farve Hvid til Næsten hvid

 

(4R,6R)-tert-butyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxan-4-acetat Anvendelse og syntese

Kemiske egenskaber hvidt til lysegult krystalpulver
Bruger

Atorvastatin mellemprodukt

(4R,6R)-6-(Cyanomethyl)-2,2-dimethyl-1,3-dioxan-4-eddikesyre 1,{{9} }Dimethylethylester er et mellemprodukt af Atorvastatin (A791750, Ca-salt), en selektiv, konkurrerende HMG-CoA-reduktase. Atorvastatin er det eneste lægemiddel i sin klasse, der er specifikt indiceret til at sænke både forhøjet LDL-kolesterol og triglyceinhibitorider hos patienter med hyperkolesterolæmi.

 

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